TD-802
TD-802 (Compound 33c) is a potent androgen receptor (AR) PROTAC degrader with high metabolic stability. It has demonstrated significant antitumor activity in vivo, supporting its use as a research tool for investigating metastatic castration-resistant prostate cancer (mCRPC) in preclinical models.
Product Specifications
CAS Number
2760703-21-5
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
CC1 (C) [C@H] (NC (=O) c2ccc (cc2) N2CCN (CC2) C2CC3 (C2) CCN (CC3) C (=O) C2CCN (CC2) c2ccc3nnn (C4CCC (=O) NC4=O) c (=O) c3c2) C (C) (C) [C@H]1Oc1ccc (C#N) c (Cl) c1
Molecular Formula
C52H61ClN10O6
Molecular Weight
957.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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