Tianeptine Metabolite MC5 sodium
MC5 is a bioactive β-oxidation metabolite of tianeptine that acts as a selective μ-opioid receptor (MOR) agonist, as demonstrated by BRET assays in HEK293T cells. Its MOR-dependent antidepressant-like efficacy is confirmed in vivo, reducing immobility in the mouse forced swim test at 30 mg/kg. This compound is a valuable research tool for studying MOR-mediated neuropharmacology and depression mechanisms.
Product Specifications
CAS Number
115220-11-6
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
O=C (CCCCNC1C2=C (N (S (=O) (C3=CC (Cl) =CC=C31) =O) C) C=CC=C2) [O-].[Na+]
Molecular Formula
C19H20ClN2O4S.Na
Molecular Weight
430.88
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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