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S1R agonist 2 hydrochloride

Compound 8b hydrochloride is a potent and selective sigma-1 receptor (S1R) agonist, exhibiting high affinity for S1R (Ki = 1.1 nM) over S2R. It has demonstrated neuroprotective properties in vitro against oxidative stress and excitotoxicity, making it a valuable tool for studying neuroprotection and neurodegenerative disease mechanisms.

Product Specifications

Field of Research

Pharmacology & Drug Discovery, Pharmacology & Drug Discovery; Cell Biology

Molecular Formula

C21H28ClNO

Molecular Weight

345.91

Storage Conditions

-20°C

Notes

For research use only.

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