VU0029251
VU0029251 is a selective mGluR5 partial antagonist with a binding affinity (Ki) of 1.07 μM. It inhibits glutamate-induced calcium mobilization in rat mGluR5-expressing cells with an IC50 of 1.7 μM, making it a useful research tool for studying neurological disorders in vitro.
Product Specifications
CAS Number
330819-85-7
Field of Research
Neuroscience
Smiles
CSC1=NC2=C (C3=C (CCC3) S2) C (N) =N1
Molecular Formula
C10H11N3S2
Molecular Weight
237.34
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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