TGR5 Receptor Agonist 4
TGR5 Receptor Agonist 4 is a potent and selective small molecule agonist for the bile acid receptor TGR5, demonstrating EC50 values of 2 nM (hTGR5) and 3 nM (mTGR5) . It is a valuable research tool for studying TGR5-mediated metabolic functions, including glucose homeostasis and body weight regulation, in both in vitro and in vivo models.
Product Specifications
CAS Number
1872436-42-4
Field of Research
Pharmacology & Drug Discovery
Smiles
C (OCC1=C (OC) C=CC=C1) (=O) C=2[C@@H] (CC (=O) N (C[C@H]3CCCO3) C2C) C=4C=CC (Cl) =NC4
Molecular Formula
C25H27ClN2O5
Molecular Weight
470.95
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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