RXFP1 receptor agonist-4
RXFP1 receptor agonist-4 (Example 268) is a potent small molecule agonist of the human RXFP1 receptor, exhibiting an EC50 of 4.9 nM for cAMP suppression in stable HEK293 cell assays. This compound is a valuable research tool for investigating relaxin receptor signaling in both cellular and animal models of fibrosis and cardiovascular disease.
Product Specifications
CAS Number
2941376-76-5
Field of Research
Pharmacology & Drug Discovery
Smiles
O=C (NC1=CC=C (F) C (=C1) C (F) (F) F) C=2SC=3C=C (C=CC3C2NC (=O) C=4C=C (C=CC4OC) C5=NOC6CC (CO) CC56) C (F) (F) F
Molecular Formula
C32H24F7N3O5S
Molecular Weight
695.6
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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