RXFP1 receptor agonist-3
Example 223 is a potent small molecule agonist of the human RXFP1 receptor with an EC50 of 2 nM, demonstrated to inhibit cAMP production in HEK293 cells. This tool compound is valuable for in vitro studies investigating relaxin signaling pathways and receptor pharmacology in cardiovascular and fibrotic disease research.
Product Specifications
CAS Number
2924767-53-1
Field of Research
Pharmacology & Drug Discovery
Smiles
C (=C/1\[C@@]2 ([C@@H] (NC (=O) C3=CC (=CC=C3OC) C4=CC (C (OC (NC5=C (F) C=CC=C5) =O) C (F) (F) F) =CC=C4F) [C@@H] (C (NC6=CC (C (F) (F) F) =C (F) C=C6) =O) [C@]1 (CC2) [H]) [H]) \C7CC7
Molecular Formula
C42H34F9N3O5
Molecular Weight
831.72
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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