RXFP1 receptor agonist-1
RXFP1 receptor agonist-1 (Example 2) is a potent small molecule agonist for the human RXFP1 receptor, demonstrating an EC50 of 300 nM for cAMP suppression in constitutively expressing HEK293 cells. This tool compound is useful for in vitro studies of relaxin signaling pathways and receptor pharmacology in metabolic and fibrotic disease research.
Product Specifications
CAS Number
2924619-64-5
Field of Research
Pharmacology & Drug Discovery
Smiles
C (NC1=CC (C (F) (F) F) =C (F) C=C1) (=O) [C@H]2[C@@]3 (\C (=C\C (F) (F) F) \[C@] ([C@H]2NC (=O) [C@H]4C[C@H] (CCC4) C5=CC (C (O) =O) =CC=C5) (CC3) [H]) [H]
Molecular Formula
C31H29F7N2O4
Molecular Weight
626.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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