Antitumor agent-101
Antitumor agent-101 is a potent and selective covalent inhibitor of the lysine methyltransferases G9a and GLP, with IC50 values of 8.5 nM and 5.5 nM, respectively. It demonstrates antitumor activity in a PANC-1 xenograft model, making it a valuable chemical probe for epigenetic cancer research in both cellular and animal studies.
Product Specifications
CAS Number
2848632-52-8
Field of Research
Epigenetics & Chromatin, Pharmacology & Drug Discovery
Smiles
N (C=1C2=C (C=C (OCCCN3CCCC3) C (OC) =C2) N=C (N (C (C=C) =O) C) N1) C4CCN (C) CC4
Molecular Formula
C26H38N6O3
Molecular Weight
482.62
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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