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GPR3 agonist-2

GPR3 agonist-2 (compound 32) is a potent and efficacious small-molecule agonist for the GPR3 receptor, demonstrating an IC50 of 260 nM. This tool compound is utilized in neuroscience research, particularly for in vitro studies investigating GPR3's role in neuronal signaling and its implications in neurodegenerative disease pathways.

Product Specifications

CAS Number

1983120-51-9

Field of Research

Pharmacology & Drug Discovery

Smiles

O=S (=O) ([O-]) C (F) (F) F.FC (F) (F) OC=1C=CC2=C ([I+]C=3C=CC=CC32) C1

Molecular Formula

C14H7F6IO4S

Molecular Weight

512.16

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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