BMS-986172
BMS-986172 is a potent and selective oral MGAT2 inhibitor with single-digit nM IC50 values. It demonstrates in vitro metabolic stability and reduces food intake and body weight in vivo, making it a valuable research tool for studying metabolic diseases such as obesity and NASH.
Product Specifications
CAS Number
1808258-99-2
Field of Research
Metabolism Research
Smiles
[C@] (F) (F) (F) [C@]1 (CC (=C (C (=O) N1) N2N=NNC2=O) C3=NN (CC4CC4) C=C3) C5=C (F) C=C (OCCCC (F) (F) F) C=C5
Molecular Formula
C24H22F7N7O3
Molecular Weight
589.47
Storage Conditions
-20°C
Notes
For research use only.
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