PF-04958242
PF-04958242 is a novel potent, selctive, and orally-active AMPA receptor (AMPAR) positive allosteric modulator (PAM) with Ki of 170 nM, EC50 of 370 nM; is under development for the treatment of cognitive symptoms in schizophrenia.Schizophrenia Phase 1 Discontinued.
Product Specifications
CAS Number
1258963-59-5
Product Name Alternative
PF04958242
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 100 mg/mL (254.78 mM)
Smiles
CC (C) S (=O) (=O) NC1COCC1OC2=CC=C (C=C2) C3=CC=C (S3) C#N
Molecular Formula
C18H20N2O4S2
Molecular Weight
392.49
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
N- ((3S,4S) -4- (4- (5-cyano-2-thienyl) phenoxy) tetrahydro-3-furanyl) -2-propanesulfonamide
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