AG 045572
AG-045572 is a potent and selective GnRH receptor antagonist with Ki values of 6.0 nM (human) and 3.8 nM (rat) . It is metabolized by CYP3A and inhibits testosterone production, making it a useful research tool for studying hormone-dependent conditions in both in vitro and in vivo models.
Product Specifications
CAS Number
263847-55-8
Product Name Alternative
GNRHReceptor, GNRH Receptor, CYP3A, AG045572, AG-045572, AG 045572
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Purity
98.99% (May vary between batches)
Solubility
DMSO:55 mg/mL (111.88 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.07 mM)
Smiles
CC1 (C) C=2C (=CC (C) =C (CC=3OC (C (NC4=C (OC) C=C (OC) C=C4OC) =O) =CC3) C2) C (C) (C) CC1
Molecular Formula
C30H37NO5
Molecular Weight
491.62
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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