ADRA1D receptor antagonist 1 free base
This potent and selective α1D-adrenoceptor antagonist (Ki = 1.6 nM) inhibits bladder contraction with an IC30 of 15 nM. It is a valuable research tool for investigating overactive bladder pathophysiology, supporting both in vitro binding assays and in vivo models of urinary urgency, frequency, and incontinence.
Product Specifications
CAS Number
1191908-24-3
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
[C@H] (C) (N1C (=N) C (C (N) =O) =CC (Cl) =C1) C2=CC (C#N) =CC=C2
Molecular Formula
C15H13ClN4O
Molecular Weight
300.74
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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