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ARTD10/PARP10-IN-2

ARTD10/PARP10-IN-2 is a dual inhibitor of mono-ADP-ribosyltransferase ARTD10/PARP10 (IC50 = 2.0 μM) and poly (ADP-ribose) polymerase-1 ARTD1/PARP1 (IC50 = 9.7 μM) . This cell-permeable compound is a valuable chemical probe for investigating ADP-ribosylation signaling in DNA damage response and cellular physiology studies in vitro.

Product Specifications

CAS Number

1708103-69-8

Field of Research

Epigenetics & Chromatin, Molecular Biology

Smiles

N (C (/C=C\C (NC) =O) =O) C1=CC (C (N) =O) =CC=C1

Molecular Formula

C12H13N3O3

Molecular Weight

247.25

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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