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BRD4 Inhibitor-26

BRD4 Inhibitor-26 is a dual-function small molecule combining BRD4 bromodomain inhibition with nitric oxide donation. It demonstrates potent activity against both BD1 and BD2 domains with IC50 values of 0.82 μM and 1.94 μM, respectively. This compound is applied in ovarian cancer research, showing utility in both in vitro cellular studies and in vivo tumor model experiments.

Product Specifications

Field of Research

Epigenetics & Chromatin, Epigenetics & Chromatin; Pharmacology & Drug Discovery

Molecular Formula

C29H27N5O6S

Molecular Weight

573.62

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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