Cavα2δ1&NET-IN-3
Cavα2δ1&NET-IN-3 (example 216) is a dual-target small molecule inhibitor of the voltage-gated calcium channel α2δ-1 subunit and the norepinephrine transporter (NET), with Ki values of approximately 100 nM and 500 nM, respectively. This compound is a useful research tool for investigating pain signaling and sympathetic nervous system function in both cellular and animal models.
Product Specifications
CAS Number
2143584-82-9
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
O=C1C=2C (=NC (NCC) =NC2) N (C) CCN1C3=CC (O[C@@H] (CCNC) C4=CC=CS4) =CC=C3
Molecular Formula
C24H30N6O2S
Molecular Weight
466.6
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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