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NSD3-IN-2

NSD3-IN-2 is a potent small molecule inhibitor of NSD3 with an IC50 of 17.97 μM. It demonstrates significant anti-proliferative activity in non-small cell lung cancer (NSCLC) cell lines such as H460, H1299, and H1650, supporting its use as a chemical probe for oncology research targeting epigenetic regulators.

Product Specifications

CAS Number

675190-57-5

Field of Research

Epigenetics & Chromatin

Smiles

C (COC=1C2=C (C=CC1) C=CC=C2) N3C=4C (NC3=S) =C (N) N=CN4

Molecular Formula

C17H15N5OS

Molecular Weight

337.4

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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