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BT-GSI

BT-GSI is a bone-targeting γ-secretase inhibitor that blocks Notch signaling. It demonstrates dual anti-myeloma and anti-resorptive activity in research, showing potential to inhibit tumor progression and osteolytic lesions in preclinical models of multiple myeloma and bone metastatic disease.

Product Specifications

Field of Research

Neuroscience, Protein Biochemistry, Stem Cell & Developmental Biology

Smiles

CC[C@H] (C) [C@@H] (C (=O) N[C@@H] (CC (C) C) /C=N/N (C) CCCC (=O) NC (P (=O) (O) O) P (=O) (O) O) NC (=O) OCC1=CC=CC=C1.Br

Molecular Formula

C26H46BrN5O10P2

Molecular Weight

730.52

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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