GPI-15427
GPI-15427 is a brain-penetrant, nanomolar-potency PARP-1 inhibitor. It enhances the efficacy of temozolomide and radiotherapy in CNS tumors and HNSCC, as demonstrated in preclinical in vitro and in vivo studies for glioblastoma and lymphoma research.
Product Specifications
CAS Number
805242-85-7
Field of Research
Epigenetics & Chromatin, Metabolism Research, Molecular Biology
Smiles
O=C1C2=C3C (C=4C (OC3=CC=C2) =CC=C (CN5CCN (C) CC5) C4) =NN1
Molecular Formula
C20H20N4O2
Molecular Weight
348.4
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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