NH2-c[X-R-L-S-X]-K-G-P- (D-1Nal)
Selected Variant
GTR19220022-01
Size: 5 mg
Compound 39 is a potent and balanced APJ receptor agonist with sub-nanomolar binding affinity (Ki = 0.6 nM) . It effectively activates Gαi1 signaling (EC50 = 0.8 nM) and recruits β-arrestin2 (EC50 = 31 nM), making it a valuable tool for studying APJ receptor pharmacology in cardiovascular research, both in vitro and in vivo.
Product Specifications
CAS Number
2891469-80-8
Field of Research
Pharmacology & Drug Discovery
Molecular Formula
C49H73N13O11
Molecular Weight
1020.18
Storage Conditions
-20°C
Notes
For research use only.
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