CMKLR1 antagonist 1
CMKLR1 antagonist 1 (S-26d) is a potent and orally bioavailable small molecule inhibitor of chemokine-like receptor 1, demonstrating a pIC50 of 7.44 in vitro using hCMKLR1-transfected CHO cells. This antagonist is a valuable research tool for studying the Chemerin/CMKLR1 axis in disease models, including psoriasis and metabolic disorders such as obesity and insulin resistance.
Product Specifications
Field of Research
Immunology & Inflammation, Infectious Disease & Virology, Pharmacology & Drug Discovery
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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