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Carboxylesterase-IN-2

Carboxylesterase-IN-2 is a potent and selective Notum carboxylesterase inhibitor with an IC50 of ≤10 nM. This compound is a valuable research tool for investigating the role of Notum in Wnt signaling pathways, with applications in cancer-related in vitro and in vivo studies.

Product Specifications

CAS Number

2764748-88-9

Product Name Alternative

Carboxylesterase, Carboxylesterase-IN-2, betacatenin, beta-catenin, 1,2,4Triazolo[4,3b]pyridazin3 (2H) one,6[ (3,4dimethylphenyl) thio], bcatenin, Wnt, Wnt/b-catenin, Wnt/betacatenin, Wnt/β-catenin, βcatenin

Field of Research

Metabolism Research, Signal Transduction, Stem Cell & Developmental Biology

Purity

99.49% (May vary between batches)

Solubility

DMSO:70 mg/mL (257.04 mM)

Smiles

O=C1N2C (C=CC (SC3=CC (C) =C (C) C=C3) =N2) =NN1

Molecular Formula

C13H12N4OS

Molecular Weight

272.33

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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