GnRH-R antagonist 1
Compound 21a is a potent, orally bioavailable GnRH receptor antagonist with high binding affinity (IC50=0.57 nM) and in vitro efficacy (IC50=2.18 nM) . It is a research tool for studying advanced prostate cancer and for the prevention of premature luteinizing hormone surges in assisted reproductive technology protocols.
Product Specifications
CAS Number
2826273-90-7
Field of Research
Pharmacology & Drug Discovery
Smiles
CN (CCOC (F) (F) F) CC1=C (SC2=C1C (=O) N (C (=O) N2CC3=C (C=CC=C3F) F) C4=NN=C (C=C4) OC) C5=CC=C (C=C5) NC (=O) NOC
Molecular Formula
C31H28F5N7O6S
Molecular Weight
721.65
Storage Conditions
-20°C
Notes
For research use only.
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