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FGFR3-IN-5

FGFR3-IN-5 is a highly selective small molecule inhibitor of FGFR3 (IC50 = 3 nM), with significantly lower activity against FGFR2 and FGFR1. It is a valuable research tool for investigating FGFR3-driven oncogenesis in both cellular assays and preclinical in vivo cancer models.

Product Specifications

CAS Number

2446664-72-6

Field of Research

Cardiovascular Research, Cell Biology, Signal Transduction

Smiles

O (C) C=1C=2N (C=C (C1) C3=CN (N=C3) C4CCN (C (=O) C5 (F) CN (C (C=C) =O) C5) CC4) N=CC2C#N

Molecular Formula

C24H24FN7O3

Molecular Weight

477.49

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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