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DC-BPi-03

DC-BPi-03 is a potent small molecule inhibitor targeting the BPTF bromodomain, exhibiting an IC50 of 698.3 nM. It demonstrates promising anticancer activity in leukemia research, suitable for both in vitro mechanistic studies and in vivo efficacy models in oncology.

Product Specifications

CAS Number

2758411-46-8

Product Name Alternative

BPTF, EpigeneticReaderDomain, Epigenetic Reader Domain

Field of Research

Epigenetics & Chromatin, Immunology & Inflammation

Purity

98.96% (May vary between batches)

Solubility

10% DMSO+40% PEG300+5% Tween 80+45% Saline:2.5 mg/mL (8.27 mM) ; DMSO:20 mg/mL (66.15 mM)

Smiles

O=S (=O) (C=1N=C (C=C (N1) C2=CC=C3NC=CC3=C2) NC) C

Molecular Formula

C14H14N4O2S

Molecular Weight

302.35

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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