DBRD4-BD1
DBRD4-BD1 is a selective BRD4 bromodomain degrader (DC50 = 280 nM) that uniquely upregulates BRD2/3, distinguishing it from pan-BET degraders. Its selectivity facilitates precise BRD4 biology studies in vitro and enables the design of novel heterobifunctional probes for targeted protein degradation research.
Product Specifications
CAS Number
2839318-19-1
Field of Research
Epigenetics & Chromatin, Immunology & Inflammation, Pharmacology & Drug Discovery
Smiles
O (C=1N=C (C2=C (N=CN2C3CCN (CCOCCOCCNC (COC4=C5C (C (=O) N (C5=O) C6C (=O) NC (=O) CC6) =CC=C4) =O) CC3) C7=CC=C (C (F) (F) F) C=C7) C=CN1) C8=CC (C (C) C) =CC=C8C
Molecular Formula
C50H53F3N8O9
Molecular Weight
967
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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