TG11-77 HCl
TG11-77 HCl is a potent, selective, and brain-permeable EP2 receptor antagonist with a Schild KB of 9.7 nM. Its favorable solubility, pharmacokinetics, and brain exposure make it a valuable second-generation tool compound for investigating EP2-mediated pathways in neurological and inflammatory disease models, both in vitro and in vivo.
Product Specifications
CAS Number
2490544-34-6
Smiles
C (CNC (=O) C=1C=NC (NC2=CC (C) =CC (C) =N2) =NC1) C=3C=4C (NC3C) =CC=CC4.Cl
Molecular Formula
C23H24N6O.xHCl
Molecular Weight
436.944
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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