GSK-2807 free base
GSK2807 is a potent, selective, and SAM-competitive SMYD3 inhibitor (Ki = 14 nM) that occupies both the cofactor and substrate-binding sites. It has demonstrated anti-proliferative effects in cancer cell lines and has been utilized as a chemical probe to investigate SMYD3's role in oncology and epigenetics research.
Product Specifications
CAS Number
2245255-65-4
Field of Research
Epigenetics & Chromatin
Smiles
O[C@H]1[C@H] (N2C=3C (N=C2) =C (N) N=CN3) O[C@H] (CN (CC[C@@H] (C (O) =O) N) CCCN (C) C) [C@H]1O
Molecular Formula
C19H32N8O5
Molecular Weight
452.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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