RK-52
RK-52 is a potent and selective synthetic inhibitor of the trypanosomal cysteine protease rhodesain, exhibiting a rapid second-order rate constant of 6.7 x 107 M−1 min−1 and sub-nanomolar affinity (Ki = 38 pM) . This inhibitor is a valuable chemical tool for studying Trypanosoma brucei biology and for anti-parasitic drug discovery research in both in vitro and in vivo experimental models.
Product Specifications
CAS Number
2127401-37-8
Smiles
[C@H] (CC1=CC=CC=C1) (C (N[C@@H] (CCC2=CC=CC=C2) /C=C/C (C) =O) =O) NC (OCC3=CC=CC=C3) =O
Molecular Formula
C30H32N2O4
Molecular Weight
484.59
Storage Conditions
-20°C
Notes
For research use only.
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