DG046
DG046 is a potent, phosphinic pseudopeptide inhibitor of ERAP1 that occupies the enzyme's active site and is stabilized by an extensive, unusual π-stacking network. This inhibitor is a valuable research tool for studying antigen processing in immunology and oncology, with utility in both in vitro enzymatic assays and cellular models.
Product Specifications
CAS Number
2007955-23-7
Smiles
[C@H] (C (N[C@@H] (CC1=CC=CC=C1) C (N) =O) =O) (CP ([C@H] (CCC2=CC=CC=C2) N) (=O) O) CC#C
Molecular Formula
C24H30N3O4P
Molecular Weight
455.49
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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