EPZ032597
EPZ032597 is a potent and selective SMYD2 inhibitor (IC50 = 16 nM) with demonstrated anticancer activity. Research indicates its utility in studying epigenetic mechanisms in oncology, showing efficacy in preclinical models of pancreatic cancer, including in vitro cell studies and in vivo tumor growth inhibition.
Product Specifications
CAS Number
1887193-58-9
Product Name Alternative
EPZ032597, EPZ-032597, EPZ 032597, Grp94-IN2, Grp94 IN 2, Grp94 IN-2, Grp94-IN 2, Grp94IN2, Histone Methyltransferase, HistoneMethyltransferase, SMYD2
Field of Research
Epigenetics & Chromatin
Purity
99.41% (May vary between batches)
Solubility
DMSO:55 mg/mL (145.72 mM)
Smiles
C (NC1CN (CC2=CN (CC3=CC=CC=C3) N=C2) C1) (=O) C4=CN (N=N4) C5CC5
Molecular Formula
C20H23N7O
Molecular Weight
377.44
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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