GAT100
GAT-100 is a covalent negative allosteric modulator (NAM) of CB1R that paradoxically enhances orthosteric agonist binding. This unique covalent probe is a valuable tool for mapping allosteric sites and investigating CB1 receptor modulation in both in vitro binding assays and cellular signaling studies.
Product Specifications
CAS Number
1663564-42-8
Smiles
C (C) C=1C=2C (NC1C (NCCC3=CC=C (C=C3) N4CCCCC4) =O) =CC=C (N=C=S) C2
Molecular Formula
C25H28N4OS
Molecular Weight
432.58
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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