ZEN-2759
ZEN-2759 is a potent and selective small molecule inhibitor targeting the bromodomains of BRD4, including BD1, BD2, and the tandem BD1BD2. It is a valuable chemical probe for BET protein research in oncology and inflammation, with utility in both in vitro biochemical assays and in vivo disease model studies.
Product Specifications
CAS Number
1616400-50-0
Product Name Alternative
BRD4 (1), BRD4 (2), CHF6366, CHF 6366, EpigeneticReaderDomain, Epigenetic Reader Domain, ZEN2759, ZEN-2759, ZEN 2759
Field of Research
Epigenetics & Chromatin
Purity
99.36% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (7.13 mM) ; DMSO:60 mg/mL (214.04 mM)
Smiles
CC=1C (C2=CN (CC3=CC=CC=C3) C (=O) C=C2) =C (C) ON1
Molecular Formula
C17H16N2O2
Molecular Weight
280.32
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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