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EPZ020809

EPZ020809 is a potent and selective small molecule inhibitor of the histone demethylase KDM4C, exhibiting a Ki of 31 nM. This compound is a valuable research tool for investigating the role of KDM4C in oncology, epigenetics, and both cellular and animal model studies.

Product Specifications

CAS Number

1503332-97-5

Smiles

C (O) (=O) C=1C=C (N=CC1) C2=CC=CN2

Molecular Formula

C10H8N2O2

Molecular Weight

188.18

Storage Conditions

-20°C

Notes

For research use only.

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