CGP 55845
CGP 55845 is a potent and selective GABAB receptor antagonist with a pKi of 8.35, effectively blocking agonist binding. It inhibits the release of GABA and glutamate, demonstrated by pEC50 values of 8.08 and 7.85, respectively. This compound is widely used in neuroscience research to study synaptic transmission and neurotransmitter release in both in vitro and in vivo models.
Product Specifications
CAS Number
150175-54-5
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
[C@H] (NC[C@@H] (CP (CC1=CC=CC=C1) (=O) O) O) (C) C2=CC (Cl) =C (Cl) C=C2
Molecular Formula
C18H22Cl2NO3P
Molecular Weight
402.25
Storage Conditions
-20°C
Notes
For research use only.
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