ML 252
ML252 is a potent and selective KCNQ2 (Kv7.2) potassium channel blocker (IC50=69 nM) and a broad cytochrome P450 inhibitor, notably of CYP3A4 (IC50=3.9 nM) . This dual pharmacological profile makes it a valuable research tool for studying neuronal excitability, drug metabolism interactions, and epilepsy mechanisms in vitro.
Product Specifications
CAS Number
1392494-64-2
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
N (C ([C@@H] (CC) C1=CC=CC=C1) =O) C2=C (C=CC=C2) N3CCCC3
Molecular Formula
C20H24N2O
Molecular Weight
308.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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