EST64454 free base
EST64454 is a potent and selective σ1 receptor antagonist clinical candidate for pain treatment. Its favorable BCS Class I profile, characterized by high solubility and Caco-2 permeability, alongside high metabolic stability, supports its utility in both in vitro mechanistic studies and in vivo pain research models.
Product Specifications
CAS Number
1351438-26-0
Field of Research
Pharmacology & Drug Discovery
Smiles
C (OCCN1CCN (C (C) =O) CC1) C2=NN (C=C2) C3=CC (F) =C (F) C=C3
Molecular Formula
C18H22F2N4O2
Molecular Weight
364.39
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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