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Famitinib malate

Famitinib malate (SHR1020) is an oral multi-targeted tyrosine kinase inhibitor with potent activity against c-kit, VEGFR-2, and PDGFRβ. It induces apoptosis and has demonstrated significant antitumor efficacy in both in vitro studies and in vivo xenograft models of gastric cancer, supporting its use in oncology research.

Product Specifications

CAS Number

1256377-67-9

Field of Research

Cardiovascular Research, Cell Biology, Signal Transduction

Smiles

[C@H] (CC (O) =O) (C (O) =O) O.C (=C\1/C=2C (NC1=O) =CC=C (F) C2) \C3=C (C) C4=C (N3) CCN (CCN (CC) CC) C4=O

Molecular Formula

C27H33FN4O7

Molecular Weight

544.57

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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