CBP/p300-IN-2
CBP/EP300-IN-2 is a potent small molecule inhibitor of the CBP and EP300 bromodomains, with IC50 values of 1.07 nM and 5.96 nM, respectively. It serves as a valuable chemical probe for epigenetic research, enabling the study of histone acetylation-dependent transcriptional regulation in both cellular and biochemical assays.
Product Specifications
CAS Number
2158265-96-2
Field of Research
Cell Biology, Epigenetics & Chromatin, Signal Transduction
Smiles
C (NC) (=O) N1CC=2C (=NN (C2CC1) C3CCOCC3) C=4C5=C (C=C (C (C (F) F) =C5) C6=CN (C) N=C6) C=NC4
Molecular Formula
C27H29F2N7O2
Molecular Weight
521.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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