CGP 20712 A
CGP 20712 A mesylate is a potent and selective β1-adrenergic receptor antagonist with an IC50 of 0.7 nM. It is utilized in cardiovascular research to study receptor function and has demonstrated in vivo activity, such as reversing gastric relaxation and lowering blood pressure in experimental models.
Product Specifications
CAS Number
105737-62-0
Product Name Alternative
AdrenergicReceptor, Adrenergic Receptor, CGP20712 Mesylate, CGP-20712 Mesylate, CGP 20712 mesylate, CGP 20712 A, β1-adrenoceptor, β1-adrenergic receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.91% (May vary between batches)
Solubility
DMSO:80 mg/mL (135.46 mM)
Smiles
O=C (N) C1=CC (OCCNCC (O) COC=2C=CC (=CC2) C3=NC (=CN3C) C (F) (F) F) =CC=C1O.O=S (=O) (O) C
Molecular Formula
C24H29F3N4O8S
Molecular Weight
590.57
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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