CPUY074020
CPUY074020 is a potent, orally bioavailable small molecule inhibitor of the histone methyltransferase G9a, exhibiting an IC50 of 2.18 μM. It demonstrates anti-proliferative activity in cellular assays and serves as a valuable chemical probe for epigenetic research in oncology and other fields involving histone methylation.
Product Specifications
CAS Number
902279-44-1
Product Name Alternative
CPUY 074020, CPUY074020, CPUY-074020, HistoneMethyltransferase, Histone Methyltransferase, G9a
Field of Research
Epigenetics & Chromatin
Purity
98.64% (May vary between batches)
Solubility
DMSO:4.17 mg/mL (10.01 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.4 mM)
Smiles
N (CCN1CCCC1) C2=C3C=4C (C (=C2) N5CCCCC5) =NOC4C=6C (C3=O) =CC=CC6
Molecular Formula
C25H28N4O2
Molecular Weight
416.52
Storage Conditions
-20°C
Notes
For research use only.
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