CSRM617
CSRM617 is a selective small molecule inhibitor of the transcription factor ONECUT2 (OC2), binding its HOX domain with a Kd of 7.43 μM. It induces apoptosis via Caspase-3 and PARP cleavage and has demonstrated good tolerability in a prostate cancer mouse model, supporting its use in oncology research.
Product Specifications
CAS Number
787504-88-5
Field of Research
Cell Biology, Metabolism Research
Smiles
C (=NNC (C (CO) N) =O) C1=C (O) C (O) =C (O) C=C1
Molecular Formula
C10H13N3O5
Molecular Weight
255.23
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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