Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

EGFR-IN-2

EGFR-IN-2 is an orally bioavailable, mutation-selective EGFR inhibitor designed for NSCLC research. It potently targets T790M resistance mutants (IC50 27-33 nM) while sparing wild-type EGFR (IC50 218 nM) . This profile supports its investigation in preclinical models for overcoming tyrosine kinase inhibitor resistance.

Product Specifications

CAS Number

1643497-70-4

Product Name Alternative

EGFRIN2, EGFR, EGFR IN 2

Field of Research

Cardiovascular Research, Cell Biology, Signal Transduction

Purity

98.52% (May vary between batches)

Smiles

[C@@H] (CC) (C) N1N=C (C=2C1=CC (NC3=NC (=NC=C3) C4=CN (S (=O) (=O) C5CC5) N=C4) =NC2) N6CC (C (C) (C) O) C6

Molecular Formula

C26H33N9O3S

Molecular Weight

551.66

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Norovirus Genogroup II discontinued, see 353487
471184 1 mg

Norovirus Genogroup II discontinued, see 353487

Sign In for Pricing
View Details
TTC39B Protein Vector (Rat) (pPB-N-His)
PV313555 500 ng

TTC39B Protein Vector (Rat) (pPB-N-His)

Sign In for Pricing
View Details
Apolipoprotein AI (Apo AI, ApoA-I, Apolipoprotein A1, APOA1) (Biotin) discontinued
A2299-12X-Biotin 5 mL

Apolipoprotein AI (Apo AI, ApoA-I, Apolipoprotein A1, APOA1) (Biotin) discontinued

Sign In for Pricing
View Details
ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)
TRV-0063403-01 24 Tests

ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)

Sign In for Pricing
View Details
ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)
TRV-0063403-02 48 Tests

ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)

Sign In for Pricing
View Details
ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)
TRV-0063403-03 96 Tests

ELISA Kit for Dihydrolipoyl Transacetylase (DLAT)

Sign In for Pricing
View Details