Elacestrant S enantiomer
The S enantiomer of Elacestrant is an orally bioavailable, selective estrogen receptor degrader (SERD) with preferential activity against ERα (IC50 = 48 nM) over ERβ (IC50 = 870 nM) . It is a research tool for investigating ER+ breast cancer mechanisms and has demonstrated antitumor efficacy in both cellular assays and in vivo xenograft models.
Product Specifications
Smiles
OC1=CC=C2C[C@@H] (C3=CC=C (OC) C=C3N (CC) CC4=CC=C (CCNCC) C=C4) CCC2=C1
Molecular Formula
C30H38N2O2
Molecular Weight
458.63
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
39737061 1.0 µg DNA
RN5S177 Lentiviral Vector (Human) (CMV) (pLenti-GIII-CMV)
Sign In for Pricing
View Details bs-9883R-BF750 100 µL
HBZ Polyclonal Antibody, AbBy Fluor™ 750 Conjugated
Sign In for Pricing
View Details 