Elacestrant S enantiomer
The S enantiomer of Elacestrant is an orally bioavailable, selective estrogen receptor degrader (SERD) with preferential activity against ERα (IC50 = 48 nM) over ERβ (IC50 = 870 nM) . It is a research tool for investigating ER+ breast cancer mechanisms and has demonstrated antitumor efficacy in both cellular assays and in vivo xenograft models.
Product Specifications
Smiles
OC1=CC=C2C[C@@H] (C3=CC=C (OC) C=C3N (CC) CC4=CC=C (CCNCC) C=C4) CCC2=C1
Molecular Formula
C30H38N2O2
Molecular Weight
458.63
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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