ERK1/2 inhibitor 1
ERK1/2 inhibitor 1 is a potent and orally active small molecule that selectively inhibits ERK1 and ERK2 with an IC50 of 3.0 nM. It is widely used in cancer research to study MAPK/ERK pathway signaling in both cellular assays and in vivo models.
Product Specifications
CAS Number
2095719-90-5
Product Name Alternative
ERK1, ERK1/2 inhibitor 1, ERK-1/2 inhibitor 1, ERK2
Field of Research
Pharmacology & Drug Discovery; Cell Biology, Signal Transduction
Purity
98.81% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (1.82 mM) ; DMSO:5.51 mg/mL (10.02 mM)
Smiles
C[C@@H] (N1Cc2ccc (cc2C1=O) -c1nc (NC2CCOCC2) ncc1Cl) C (=O) N[C@H] (CO) c1cccc (C) c1
Molecular Formula
C29H32ClN5O4
Molecular Weight
550.05
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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