GB-110
GB-110 is a potent, nonpeptidic, and orally active agonist of protease-activated receptor 2 (PAR2), selectively inducing PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. It is a valuable research tool for studying PAR2 signaling in inflammation, pain, and cancer, applicable in both in vitro and in vivo models.
Product Specifications
CAS Number
1252806-70-4
Field of Research
Pharmacology & Drug Discovery
Smiles
[C@H] (CC1CCCCC1) (C (N[C@H] (C (NCC2=CC (C (=O) N3CCC (CN) CC3) =CC=C2) =O) [C@H] (CC) C) =O) NC (=O) C4=CC=NO4
Molecular Formula
C33H48N6O5
Molecular Weight
608.77
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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