J-2156
J-2156 is a potent and selective somatostatin SST4 receptor agonist, exhibiting IC50 values of 0.05 nM (human) and 0.07 nM (rat) . In rat models of neuropathic pain, it alleviates mechanical allodynia and hyperalgesia with ED50 values of 3.7 and 8.0 mg/kg, respectively, supporting its use in pain research.
Product Specifications
CAS Number
848647-56-3
Field of Research
Pharmacology & Drug Discovery
Smiles
S (N[C@H] (C (N[C@@H] (CC1=CC=CC=C1) C (N) =O) =O) CCN) (=O) (=O) C=2C3=C (C (C) =CC2) C=CC=C3
Molecular Formula
C24H28N4O4S
Molecular Weight
468.57
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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