L-803087
L-803087 is a highly selective sst4 receptor agonist (Ki = 0.7 nM) with over 280-fold selectivity. It potentiates AMPA-mediated synaptic responses in hippocampal studies in vitro and has been shown to exacerbate seizures in alginate-induced seizure models in vivo, supporting its use in neuroscience research.
Product Specifications
CAS Number
217480-26-7
Product Name Alternative
L 803087, L803087, L-803087, sst5 receptor, sst2 receptor, sst3 receptor, sst4 receptor, SST1, sst1 receptor
Field of Research
Pharmacology & Drug Discovery
Purity
97.58% (May vary between batches)
Solubility
DMSO:55 mg/mL (113.28 mM)
Smiles
COC (=O) [C@H] (CCCNC (N) =N) NC (=O) CCCc1c ([nH]c2c (F) cc (F) cc12) -c1ccccc1
Molecular Formula
C25H29F2N5O3
Molecular Weight
485.53
Storage Conditions
-20°C
Notes
For research use only.
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